Quassinoid substances found in herbs such as tongkat ali
Quassinoids from Eurycoma
longifolia.
J Nat Prod. 2009 Dec; Miyake K, Tezuka Y, Awale S, Li F, Kadota S. Institute of
Natural Medicine, University of Toyama, 2630 Sugitani, Toyama 930-0194, Japan.
Ten new structurally diverse quassinoids (1-10) and 14 known compounds were
isolated from the stems of Eurycoma longifolia. The new compounds were two
eurycomanone-type C(20) quassinoids (1, 2), one klaineanone-type C(20)
quassinoid (3), one C(19) quassinoid (4) with a
1,2-seco-1-nor-6(5-->10)-abeo-picrasan-2,5-olide skeleton, and six
eurycomalactone-type C(19) quassinoids (5-10). Compounds 5 and 6 both possessed
a 3,4-epoxy group observed for the first time in eurycomalactones. Compound 1
had an alpha-oriented OH group at C-14 that had not been reported previously in
eurycomanone-type quassinoids. All of the isolates were evaluated for
cytotoxicity toward the highly metastatic HT-1080 human fibrosarcoma cell line,
and compounds 11, 23, and 24 showed potent cytotoxicity
Antimalarial activity of simalikalactone E, a new quassinoid from Quassia
amara L. (Simaroubaceae).
Antimicrob Agents Chemother. 2009 Oct; Cachet N, Hoakwie F, Bertani S, Bourdy G,
Deharo E, Stien D, Houel E, Gornitzka H, Fillaux J, Chevalley S, Valentin A,
Jullian V. Laboratoire de Pharmacochimie des Substances Naturelles et
Pharmacophores Redox, UMR 152, UPS, Université de Toulouse, 118 Route de
Narbonne, F-31062 Toulouse Cedex 9, France.
Evaluation of efficacy of bruceine A, a natural quassinoid compound extracted
from a medicinal plant, Brucea javanica, for canine babesiosis.
J Vet Med Sci. 2009 Jan; Nakao R, Mizukami C, Kawamura Y, Subeki, Bawm S,
Yamasaki M, Maede Y, Matsuura H, Nabeta K, Nonaka N, Oku Y, Katakura K.
Laboratory of Parasitology, Department of Disease Control, Graduate School of
Veterinary Medicine, Hokkaido University, Kita 18, Nishi 8, Sapporo, Japan.